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SM 16
CAS No. 614749-78-9
SM 16 ( —— )
产品货号. M19909 CAS No. 614749-78-9
SM 16 is a ALK5/ALK4 kinase inhibitor (Ki: 10/1.5 nM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥721 | 有现货 |
|
| 10MG | ￥1256 | 有现货 |
|
| 25MG | ￥2252 | 有现货 |
|
| 50MG | ￥3645 | 有现货 |
|
| 100MG | ￥5370 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称SM 16
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述SM 16 is a ALK5/ALK4 kinase inhibitor (Ki: 10/1.5 nM).
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产品描述SM 16 is a ALK5/ALK4 kinase inhibitor (Ki: 10/1.5 nM).
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同义词——
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通路Angiogenesis
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靶点ALK
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受体ALK4; ALK5
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研究领域Cancer
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适应症Cancer
化学信息
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CAS Number614749-78-9
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分子量430.5
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分子式C25H26N4O3
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纯度>98% (HPLC)
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溶解度DMSO: 60 mg/mL
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SMILESCc1cccc(n1)-c1[nH]c(nc1-c1ccc2OCOc2c1)C12CCC(CC1)(CC2)C(N)=O
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化学全称4-[4-(13-Benzodioxol-5-yl)-5-(6-methyl-2-pyridinyl)-1H-imidazol-2-yl]-bicyclo[2.2.2]octane-1-carboxamide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Suzuki E et al. A novel small-molecule inhibitor of transforming growth factor beta type I receptor kinase (SM16) inhibits murine mesothelioma tumor growth in vivo and prevents tumor recurrence after surgical resection. Cancer Res. 2007 Mar 1;67(5):2351-9.
产品手册
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